Chlorpheniramine

Chlorpheniramine

SCHEMBL4220

CN(C)CC[C@H](c1ccc(Cl)cc1)c1ccccn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Chlorpheniramine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 5/20 1.00
CHRM2 P08172 6/20 1.00
SLC6A2 P23975 6/20 1.00
SLC6A4 P31645 6/20 1.00
SLC6A3 Q01959 5/20 1.00
KCNH2 Q12809 5/20 1.00
HRH3 Q9Y5N1 5/20 1.00
CHRM1 P11229 4/20 1.00
ADRA2B P18089 4/20 1.00
HTR2A P28223 3/20 1.00
SCN1A P35498 3/20 1.00
SCN2A Q99250 3/20 1.00
SCN3A Q9NY46 3/20 1.00
CYP2D6 P10635 3/20 1.00
CHRM5 P08912 2/20 1.00
HRH2 P25021 2/20 1.00
NFKB1 P19838 2/20 1.00
THPO P40225 2/20 1.00
HTR2C P28335 2/20 1.00
TSHR P16473 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dexchlorpheniramine SCHEMBL3538 1.00 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL4314182 1.00 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL20956397 1.00 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL4219 1.00 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL29687335 1.00 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL5022351 0.99 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL14879822 0.99 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL506017 0.99 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL10622596 0.99 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL14879823 0.99 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 41854 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116898754-B Composition for water-based cosmetic, essence containing composition and preparation method of essence Ma Yinglong health Co.,Ltd. (CN) 2026-05-26 CN claimed
CN-122076970-A Platinum iridium bimetallic nano-enzyme, preparation method and application thereof in immunochromatography detection 2026-05-26 CN claimed
CN-122075378-A Antioxidant composition and application thereof 2026-05-26 CN claimed
CN-122072257-A Method for rapidly detecting poison in blood 中国科学院大连化学物理研究所 2026-05-22 CN claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
WO-2026102563-A1 DISUBSTITUTED PYRIMIDOPYRROLE ANALOG AND USE THEREOF 深圳湾实验室坪山生物医药研发转化中心 2026-05-21 WO claimed
US-12629422-B2 Agave syrup formulation or suspension for active pharmaceutical agents GENEXA INC. (US) 2026-05-19 US claimed
CN-122056798-A Skin care product composition containing deep seawater mineral powder and preparation method and application thereof 后羿生物医药(杭州)有限公司 2026-05-19 CN claimed
CN-122031343-A Composition with pouch removing effect, eye cream containing composition and preparation method of eye cream 马应龙大健康有限公司 2026-05-15 CN claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-4278679-A ANTIHISTAMINE, PREVENTION OF ANTICHOLINERGIC EFFECT CHROMALLOY AMERICAN CORPORATION (US) 1981-07-14 US claimed
US-4269835-A Nasal composition for relieving nasal distress WHITTLE BARRY J 1981-05-26 US claimed
US-4256763-A ANTIINFLAMMATORY AGENTS, VIRICIDES, PHENOLPHTHALEIN MCHUGH JOHN E 1981-03-17 US claimed
US-4234566-A Antihistamine and methods for use thereof CARTER-WALLACE, INC. 1980-11-18 US claimed
US-4232002-A Procedures and pharmaceutical products for use in the administration of antihistamines THE WELSH NATIONAL SCHOOL OF MEDICINE (GB) 1980-11-04 US claimed
US-4226850-A ANTIHISTAMINES CARTER-WALLACE, INC., A CORP. OF DE 1980-10-07 US claimed
US-4205060-A Microcapsules containing medicament-polymer salt having a water-insoluble polymer sheath, their production and their use PENNWALT CORPORATION (US) 1980-05-27 US claimed
US-4175119-A Composition and method to prevent accidental and intentional overdosage with psychoactive drugs PORTER GARRY L 1979-11-20 US claimed
US-4104382-A (((THIAZOLYL-, ISOTHIAZOLYL- OR PYRIDYLALKYL)THIO)ALKYL)GUANIDINE SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1978-08-01 US claimed
US-4000302-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1976-12-28 US claimed