SCHEMBL14883271

SCHEMBL14883271

CNC(=O)c1cc2ccccc2cn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.56
CYP1A2 P05177 2/20 0.54
KDM4E B2RXH2 1/20 0.54
NPC1 O15118 1/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.54
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.54
PKM P14618 1/20 0.54
HPGD P15428 1/20 0.54
TSHR P16473 1/20 0.54
APEX1 P27695 1/20 0.54
CYP2C19 P33261 1/20 0.54
THPO P40225 1/20 0.54
RAB9A P51151 1/20 0.54
PMP22 Q01453 1/20 0.54
HSD17B10 Q99714 1/20 0.54
EGFR P00533 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14876092 0.84 EGLN1 (0.57) EGLN1EGFRHDAC3HDAC1HDAC2
SCHEMBL213288 0.82 EGLN1 (0.60) EGLN1CYP1A2ALDH1A1CYP3A4MAPT
SCHEMBL15610421 0.81 KDR (0.45) CYP1A2KDM4ENPC1ALDH1A1LMNA
SCHEMBL16307678 0.81 HDAC3 (0.57) EGLN1RAB9AEGFRHDAC3HDAC1
SCHEMBL14885756 0.81 EGLN1 (0.56) EGLN1EGFRHDAC3HDAC1HDAC2
SCHEMBL8432118 0.81 EGLN1 (0.52) EGLN1ALDH1A1LMNAEGFRHDAC3
SCHEMBL29431793 0.81 EGFR (0.46) EGLN1CYP1A2KDM4ENPC1ALDH1A1
SCHEMBL15610991 0.80 PLK1 (0.61) CYP1A2KDM4ENPC1ALDH1A1LMNA
SCHEMBL29812173 0.80 PLK1 (0.61) CYP1A2KDM4ENPC1ALDH1A1LMNA
SCHEMBL5162848 0.80 EGLN1 (0.51) EGLN1CYP1A2KDM4EALDH1A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12486251-B2 CBP/EP300 inhibitor and use thereof PHARMABLOCK SCIENCES (NANJING) , INC. (CN) 2025-12-02 US disclosed
US-20230159497-A1 CBP/EP300 INHIBITOR AND USE THEREOF PHARMABLOCK SCIENCES (NANJING) , INC. (CN) 2023-05-25 US disclosed
EP-4140996-A1 CBP/EP300 INHIBITOR AND USE THEREOF PHARMABLOCK SCIENCES (NANJING), INC. (CN) 2023-03-01 EP disclosed
US-20160297763-A1 Heteroaryl hydroxamic acid derivatives and their use in the treatment, amelioration or prevention of a viral disease F. HOFFMANN-LA ROCHE LTD (CH) 2016-10-13 US disclosed
EP-2829535-A1 Intercalating amino acids Universität Konstanz (DE) 2015-01-28 EP disclosed
US-20130102600-A1 Heteroaryl hydroxamic acid derivatives and their use in the treatment, amelioration or prevention of a viral disease F. HOFFMANN-LA ROCHE LTD (CH) 2013-04-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160297763-A1 Heteroaryl hydroxamic acid derivatives and their use in the treatment, amelioration or prevention of a viral disease ALAD, CYP27A1, FAH EGLN1 1937/4885CYP1A2 226/4885KDM4E 3498/4885
US-20230159497-A1 CBP/EP300 INHIBITOR AND USE THEREOF EP300, CREBBP, BPTF EGLN1 571/4885CYP1A2 3865/4885KDM4E 440/4885
US-12486251-B2 CBP/EP300 inhibitor and use thereof EP300, CREBBP, BPTF EGLN1 571/4885CYP1A2 3865/4885KDM4E 440/4885
US-20130102600-A1 Heteroaryl hydroxamic acid derivatives and their use in the treatment, amelioration or prevention of a viral disease FAH, SLC10A1, OAT EGLN1 1655/4885CYP1A2 410/4885KDM4E 3710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.