SCHEMBL14899751

SCHEMBL14899751

NC(=O)c1cccc(CS)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ABCB11 O95342 1/20 0.40
LMNA P02545 1/20 0.40
PTGS1 P23219 1/20 0.40
ADORA1 P30542 1/20 0.40
PTGS2 P35354 1/20 0.40
FOLH1 Q04609 1/20 0.39
METAP2 P50579 1/20 0.38
GAA P10253 1/20 0.38
G6PD P11413 1/20 0.37
CASP7 P55210 1/20 0.37
CASP6 P55212 1/20 0.37
BCAT2 O15382 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8943463 0.84 ABCB11 (0.45) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL5545298 0.82 PARP1 (0.46) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL3622854 0.82 PARP1 (0.47) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL7416478 0.82 KDM4E (0.50) KDM4EALDH1A1MAPTHPGDTSHR
Ammonia Solution, Strong SCHEMBL17727872 0.81 PARP1 (0.46) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL3829415 0.79 KDM4E (0.44) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL40536 0.79 ALDH1A1 (0.54) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL5685695 0.78 MAPT (0.42) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL18426587 0.78 KDM4E (0.38) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL30742732 0.78 MAPT (0.42) KDM4EALDH1A1MAPTHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2586778-A2 Pyridazinone derivatives useful as glucan synthase inhibitors Merck Sharp & Dohme Corp. (US) 2013-05-01 EP disclosed