SCHEMBL14899790

SCHEMBL14899790

Nc1c(CSO)ccc2c1CCCN2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIA3 P42263 1/20 0.37
GRIA4 P48058 1/20 0.37
PSMB5 P28074 1/20 0.34
BCHE P06276 1/20 0.34
KDM4E B2RXH2 3/20 0.32
MAPT P10636 3/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
NUDT1 P36639 1/20 0.31
ALDH1A1 P00352 2/20 0.30
TP53 P04637 2/20 0.30
GAA P10253 2/20 0.30
ALOX15 P16050 2/20 0.30
HTT P42858 2/20 0.30
HSD17B10 Q99714 2/20 0.30
TDP1 Q9NUW8 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14080970 0.76 GRIA1 (0.40) GRIA1GRIA2GRIA3GRIA4PSMB5
SCHEMBL6780467 0.73 GRIA1 (0.45) GRIA1GRIA2GRIA3GRIA4BCHE
SCHEMBL4929162 0.70 GRIA1 (0.55) GRIA1GRIA2GRIA3GRIA4PSMB5
SCHEMBL5816157 0.68 GRIA1 (0.41) GRIA1GRIA2GRIA3GRIA4BCHE
SCHEMBL6783794 0.65 GRIA1 (0.41) GRIA1GRIA2GRIA3GRIA4BCHE
SCHEMBL7039122 0.63 NOTUM (0.46) GRIA1GRIA2GRIA3GRIA4BCHE
SCHEMBL2269074 0.63 NUDT1 (0.46) GRIA1GRIA2GRIA3GRIA4BCHE
SCHEMBL29805885 0.63 NUDT1 (0.46) GRIA1GRIA2GRIA3GRIA4BCHE
SCHEMBL3502666 0.62 CHRNE (0.41) GRIA1GRIA2GRIA3GRIA4PSMB5
SCHEMBL21187595 0.60 GRIA1 (0.46) GRIA1GRIA2GRIA3GRIA4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2586778-A2 Pyridazinone derivatives useful as glucan synthase inhibitors Merck Sharp & Dohme Corp. (US) 2013-05-01 EP disclosed