SCHEMBL14907343

SCHEMBL14907343

CCCCCCCCOc1ccc2[nH]cc(CCNC(=O)OC(C)(C)C)c2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.66
HTR1D P28221 8/20 0.66
HTR1B P28222 8/20 0.66
MAPT P10636 2/20 0.61
MAPK1 P28482 2/20 0.61
TDP1 Q9NUW8 2/20 0.61
KDM4E B2RXH2 1/20 0.61
TP53 P04637 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
HTR2A P28223 1/20 0.61
CYP2C19 P33261 1/20 0.61
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
MTNR1A P48039 8/20 0.59
MTNR1B P49286 7/20 0.59
LTA4H P09960 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14907340 1.00 HTR1A (0.66) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL8626639 0.95 HTR1A (0.59) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL8624581 0.92 MTNR1A (0.57) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL8629672 0.92 MTNR1A (0.65) HTR1AHTR1DHTR1BTDP1KDM4E
SCHEMBL8626837 0.91 HTR1A (0.65) HTR1AHTR1DHTR1BTDP1KDM4E
SCHEMBL8881982 0.91 MTNR1A (0.58) HTR1AHTR1DHTR1BTDP1KDM4E
SCHEMBL8880875 0.90 MTNR1A (0.59) HTR1AHTR1DHTR1BTDP1KDM4E
SCHEMBL8624381 0.90 HTR1A (0.63) HTR1AHTR1DHTR1BTDP1KDM4E
SCHEMBL8880324 0.89 MTNR1A (0.60) HTR1AHTR1DHTR1BTDP1KDM4E
SCHEMBL2536092 0.89 MTNR1A (0.55) HTR1AHTR1DHTR1BMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013063492-A1 NOVEL COMPOSITIONS AND METHODS FOR TREATING CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-02 WO disclosed