SCHEMBL1490977

SCHEMBL1490977

Fc1[c]ccc(-c2ccc(Cl)cc2)c1F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.35
CYP1A2 P05177 1/20 0.33
PTGS2 P35354 3/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
LMNA P02545 1/20 0.32
CYP2A6 P11509 1/20 0.32
TDO2 P48775 1/20 0.32
NR4A2 P43354 2/20 0.31
PTGS1 P23219 1/20 0.31
MAOB P27338 1/20 0.31
NOTUM Q6P988 1/20 0.31
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4372720 0.83 TDO2 (0.33) PTGS2NPC1RAB9ATDO2NR4A2
SCHEMBL1490906 0.80 ALDH1A1 (0.33) CYP2A6
SCHEMBL7808119 0.79 ALOX5AP (0.36) HSD17B10CYP2A6
SCHEMBL6797075 0.79
SCHEMBL16564208 0.78 NOTUM (0.34) MAOBNOTUM
SCHEMBL433163 0.76 CYP1A2 (0.38) AHRCYP1A2PTGS2NPC1TP53
SCHEMBL17514854 0.76 GRM2 (0.38)
SCHEMBL28172842 0.76 LMNA (0.35) CYP1A2NPC1TP53RAB9ASMN1; SMN2
SCHEMBL28172836 0.73 MPL (0.34) NPC1TP53RAB9ASMN1; SMN2HSD17B10
SCHEMBL5646728 0.72 AHR (0.43) AHRCYP1A2PTGS2LMNACYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2477982-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2012-07-25 EP disclosed
WO-2011034962-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-03-24 WO disclosed
EP-2200607-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2010-06-30 EP disclosed
WO-2009035818-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2009-03-19 WO disclosed