SCHEMBL14917042

SCHEMBL14917042

CC(C)(C)C(CC1=NN(CCC2CCCC2)C(=O)C1)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.35
ALDH1A1 P00352 4/20 0.32
TP53 P04637 1/20 0.32
DGAT1 O75907 1/20 0.32
CPB1 P15086 1/20 0.31
CPB2 Q96IY4 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KMT2A Q03164 1/20 0.31
KLK7 P49862 1/20 0.31
CNR2 P34972 2/20 0.30
CNR1 P21554 1/20 0.30
EDNRB P24530 1/20 0.30
EDNRA P25101 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15344569 0.95 RORC (0.30) RORC
SCHEMBL14916695 0.91 CNR1 (0.35) RORCCNR2CNR1EDNRBEDNRA
SCHEMBL14917349 0.90 CNR1 (0.36) RORCALDH1A1TP53DGAT1CPB2
SCHEMBL14916450 0.89 CNR1 (0.33) CPB2CNR2CNR1
SCHEMBL14916721 0.86 CNR1 (0.30) CNR2CNR1
SCHEMBL14916520 0.84 ALDH1A1 (0.31) ALDH1A1
SCHEMBL14916979 0.83 ALDH1A1 (0.44) ALDH1A1
SCHEMBL14917270 0.81
SCHEMBL14916757 0.81
SCHEMBL14916432 0.81 ALDH1A1 (0.48) ALDH1A1TP53CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8569353-B2 Pyrazole compound DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2013-10-29 US disclosed
US-20130116296-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2013-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116296-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A RORC 657/4885ALDH1A1 2035/4885TP53 4790/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.