SCHEMBL14917577

SCHEMBL14917577

Cc1cc(Cc2ccccc2)[nH]c(=O)c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.62
ADORA1 P30542 1/20 0.50
GPR84 Q9NQS5 4/20 0.47
DAO P14920 2/20 0.47
PARP1 P09874 1/20 0.46
POLB P06746 1/20 0.46
IDH1 O75874 2/20 0.46
GSK3B P49841 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
RECQL P46063 1/20 0.43
CAPN1 P07384 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11858938 0.84 GPR84 (0.68) GPR84DAO
SCHEMBL17206126 0.80 GPR84 (0.73) SMN1; SMN2GPR84
SCHEMBL1287276 0.79 SMN1; SMN2 (0.69) SMN1; SMN2ADORA1GPR84DAOPARP1
Dimethylamine SCHEMBL27691701 0.79 SMN1; SMN2 (0.63) SMN1; SMN2ADORA1GPR84DAOPARP1
SCHEMBL6613866 0.77 SMN1; SMN2 (0.57) SMN1; SMN2ADORA1GPR84DAOPARP1
Benzylthiouracil SCHEMBL815137 0.76 SMN1; SMN2 (1.00) SMN1; SMN2ADORA1GPR84DAOPARP1
SCHEMBL28487811 0.76 KMT2A (0.43) SMN1; SMN2ADORA1DAOPARP1CYP1A2
SCHEMBL9286770 0.75 PARP1 (0.51) SMN1; SMN2ADORA1DAOPARP1CAPN1
SCHEMBL28747205 0.75 SMN1; SMN2 (0.53) SMN1; SMN2GPR84DAOPARP1CAPN1
SCHEMBL27893019 0.74 SMN1; SMN2 (0.49) SMN1; SMN2ADORA1DAOPOLBIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104039956-A Method of treatment GLAXOSMITHKLINE IP NO 2 LTD 2014-09-10 CN disclosed
CN-102970869-B Indoles GLAXOSMITHKLINE LLC 2014-07-16 CN disclosed
WO-2013067300-A1 METHOD OF TREATMENT GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2013-05-10 WO disclosed
WO-2013067302-A1 METHOD OF TREATMENT GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2013-05-10 WO disclosed
CN-102970869-A Indoles GLAXOSMITHKLINE LLC 2013-03-13 CN disclosed