SCHEMBL14922248

SCHEMBL14922248

CCCOc1c(F)cc(N2CCNCC2)cc1F

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 7/20 0.45
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
HRH4 Q9H3N8 1/20 0.39
CHRNB2 P17787 3/20 0.39
CHRNA4 P43681 3/20 0.39
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
RIPK2 O43353 3/20 0.38
NOD2 Q9HC29 3/20 0.38
ACVR1 Q04771 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14922726 0.87 CHRNB2 (0.51) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4939296 0.79 ADRB1 (0.61) ADRB1CHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL11551319 0.78 ADRB1 (0.60) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL24592792 0.76 ADRB1 (0.45) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL17431869 0.76 ALDH1A1 (0.43) ADRB1CHRNB2CHRNA4
SCHEMBL8811069 0.73 ADRB1 (0.62) ADRB1CHRNB2CHRNA4HTR3EHTR3B
SCHEMBL11544382 0.73 ADRB1 (0.65) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4940896 0.73 ADRB1 (0.53) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL6416173 0.73 ADRB1 (0.55) ADRB1CHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL20139467 0.71 ADRB1 (0.53) ADRB1CHRM2CHRM4CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed