SCHEMBL14922286

SCHEMBL14922286

CN1CCN(c2ccc3c(c2)OCCO3)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.59
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
DRD2 P14416 5/20 0.56
DRD3 P35462 5/20 0.56
HTR1A P08908 1/20 0.56
ADRA2A P08913 1/20 0.56
ADRA2C P18825 1/20 0.56
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
ADRA1B P35368 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
DRD4 P21917 4/20 0.55
HTT P42858 2/20 0.53
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
HPGD P15428 1/20 0.51
BRD4 O60885 2/20 0.50
HTR3A P46098 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20907320 0.94 NPC1 (0.54) SMN1; SMN2NPC1RAB9ADRD2DRD3
SCHEMBL13727501 0.89 NPC1 (0.59) SMN1; SMN2NPC1RAB9AADRA2CHTT
SCHEMBL15981859 0.80 DRD2 (0.52) SMN1; SMN2NPC1RAB9ADRD2DRD3
SCHEMBL15981860 0.80 DRD2 (0.52) SMN1; SMN2NPC1RAB9ADRD2DRD3
SCHEMBL7503757 0.79 TGFBR1 (0.55) DRD2DRD3HTR1AADRA2AADRA2C
SCHEMBL20000624 0.78 DRD2 (0.50) SMN1; SMN2NPC1RAB9ADRD2DRD3
SCHEMBL23646854 0.77 MAPT (0.57) SMN1; SMN2NPC1RAB9ADRD2DRD3
Hydrochloric Acid SCHEMBL10407803 0.77 TGFBR1 (0.54) DRD2DRD3HTR1AADRA2AADRA2C
SCHEMBL7956979 0.77 DRD2 (0.50) NPC1RAB9ADRD2DRD3HTR1A
SCHEMBL30061277 0.77 MAPT (0.57) SMN1; SMN2NPC1RAB9ADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed