SCHEMBL1492967

SCHEMBL1492967

Cc1cc(-c2ccc(NC(=O)NCCc3ccc(Cl)cn3)cc2)ccn1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 9/20 0.55
PSEN1 P49768 3/20 0.54
PSEN2 P49810 3/20 0.54
APH1B Q8WW43 3/20 0.54
NCSTN Q92542 3/20 0.54
APH1A Q96BI3 3/20 0.54
PSENEN Q9NZ42 3/20 0.54
MAPK1 P28482 2/20 0.52
WNT3A P56704 2/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
WDR5 P61964 1/20 0.47
KDM4E B2RXH2 1/20 0.46
PORCN Q9H237 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1492798 0.86 PSEN1 (0.72) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1493027 0.84 CNR1 (0.69) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492980 0.82 MAPK1 (0.54) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492760 0.81 CNR1 (0.66) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492982 0.81 CNR1 (0.63) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492961 0.80 WNT3A (0.50) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1493021 0.79 CNR1 (0.60) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492849 0.78 WNT3A (0.55) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492676 0.78 CNR1 (0.58) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492815 0.77 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300427-A1 UREA COMPOUNDS AS GAMMA SECRETASE MODULATORS AMGEN INC. (US) 2011-03-30 EP claimed
WO-2009137404-A1 UREA COMPOUNDS AS GAMMA SECRETASE MODULATORS AMGEN INC. (US) 2009-11-12 WO claimed