SCHEMBL14933786

SCHEMBL14933786

O=C(O)N1CC2(CCN2c2ncccn2)C1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.51
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 9/20 0.40
ALDH1A1 P00352 9/20 0.40
CYP1A2 P05177 7/20 0.40
CYP3A4 P08684 7/20 0.40
CYP2C9 P11712 6/20 0.40
HPGD P15428 5/20 0.40
USP2 O75604 1/20 0.40
CYP2D6 P10635 6/20 0.40
CYP2C19 P33261 7/20 0.39
TSHR P16473 3/20 0.39
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
MAPK1 P28482 2/20 0.38
HIF1A Q16665 1/20 0.37
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23108171 0.75 GPR119 (0.52) EPHX2MEN1KMT2AHSD17B10ALDH1A1
SCHEMBL23108170 0.71 GPR119 (0.51) EPHX2HSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL29090664 0.71 PANK3 (0.40) EPHX2MEN1KMT2AHSD17B10ALDH1A1
SCHEMBL484881 0.70 MEN1 (0.66) MEN1KMT2AHSD17B10ALDH1A1CYP1A2
SCHEMBL2856220 0.68 GAA (0.61) MEN1KMT2AHSD17B10ALDH1A1CYP2C19
SCHEMBL23107920 0.67 CYP2D6 (0.47) EPHX2MEN1KMT2AHSD17B10ALDH1A1
SCHEMBL14891885 0.64 EPHX2 (0.64) EPHX2MEN1KMT2AALDH1A1CYP3A4
SCHEMBL3076557 0.63 KDM4E (0.56) MEN1KMT2AHSD17B10ALDH1A1CYP2C19
SCHEMBL9934845 0.62 GRIN1 (0.57) HSD17B10ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL23107924 0.61 ALDH1A1 (0.44) MEN1KMT2AHSD17B10ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013064467-A1 AZETIDINE COMPOUNDS, COMPOSITIONS AND THEIR USE AS INHIBITORS OF SOLUBLE EPOXIDE HYDROLASE F. HOFFMANN-LA ROCHE AG (CH) 2013-05-10 WO disclosed