SCHEMBL14935010

SCHEMBL14935010

COB(OC)c1ccc2[nH]ncc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.49
NOS1 P29475 4/20 0.49
ROCK1 Q13464 2/20 0.49
MAPT P10636 2/20 0.49
RAB9A P51151 2/20 0.49
METAP2 P50579 1/20 0.49
CSNK2A1 P68400 1/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
KMT2A Q03164 1/20 0.49
HIF1A Q16665 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
GSK3B P49841 3/20 0.45
CLK1 P49759 2/20 0.45
DYRK3 O43781 1/20 0.45
CLK2 P49760 1/20 0.45
CLK3 P49761 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29636278 0.77 ROCK2 (0.53) ROCK2NOS1ROCK1MAPTRAB9A
SCHEMBL481818 0.77 ROCK2 (0.53) ROCK2NOS1ROCK1MAPTRAB9A
Hydrochloric Acid SCHEMBL29957203 0.75 ROCK2 (0.52) ROCK2NOS1ROCK1MAPTRAB9A
SCHEMBL1141784 0.73 RAB9A (0.57) ROCK2NOS1ROCK1MAPTRAB9A
SCHEMBL14983547 0.71 TUBB4A (0.47) MAPTRAB9AMEN1GAAKMT2A
SCHEMBL8835 0.70 ROCK1 (0.41) ROCK2NOS1ROCK1MAPTRAB9A
SCHEMBL348190 0.70 NPC1 (0.58) ROCK2ROCK1RAB9AMEN1KMT2A
SCHEMBL29643714 0.70 NPC1 (0.58) ROCK2ROCK1RAB9AMEN1KMT2A
SCHEMBL29409358 0.70 ROCK2 (0.59) ROCK2NOS1ROCK1MAPTRAB9A
SCHEMBL12872 0.70 ROCK2 (0.59) ROCK2NOS1ROCK1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110357813-A A kind of new indole amine 2,3- dioxygenase inhibitor and its preparation method and application 信达生物制药(苏州)有限公司 2019-10-22 CN disclosed
WO-2013064445-A1 IMIDAZOPYRIDAZINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2013-05-10 WO disclosed