SCHEMBL14935501

SCHEMBL14935501

CC1(CCc2ccc(O)cc2)NC(=O)NC1=O

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.68
NPSR1 Q6W5P4 1/20 0.68
ALDH1A1 P00352 3/20 0.51
MMP2 P08253 5/20 0.45
MMP9 P14780 1/20 0.45
HSD17B10 Q99714 1/20 0.45
FPR2 P25090 2/20 0.44
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
AKR1B1 P15121 1/20 0.41
ADAMTS5 Q9UNA0 7/20 0.40
ATM Q13315 1/20 0.40
MMP13 P45452 3/20 0.39
ADAMTS4 O75173 2/20 0.39
MMP3 P08254 1/20 0.39
MMP12 P39900 1/20 0.39
LMNA P02545 1/20 0.38
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14935402 1.00 SMN1; SMN2 (0.68) SMN1; SMN2NPSR1ALDH1A1MMP2MMP9
SCHEMBL14935536 0.84 SMN1; SMN2 (0.68) SMN1; SMN2NPSR1ALDH1A1MMP2MMP9
SCHEMBL12378835 0.84 SMN1; SMN2 (0.68) SMN1; SMN2NPSR1ALDH1A1MMP2FPR2
SCHEMBL9584263 0.83 SMN1; SMN2 (0.68) SMN1; SMN2NPSR1ALDH1A1MMP2MMP9
SCHEMBL12378834 0.78 SMN1; SMN2 (0.60) SMN1; SMN2NPSR1ALDH1A1MMP2ADAMTS5
SCHEMBL11767593 0.78 SMN1; SMN2 (0.53) SMN1; SMN2NPSR1ALDH1A1MMP2HSD17B10
SCHEMBL11701498 0.75 SMN1; SMN2 (0.50) SMN1; SMN2NPSR1ALDH1A1MMP2ADAMTS5
SCHEMBL11700800 0.75 NPSR1 (0.50) SMN1; SMN2NPSR1ALDH1A1MMP2ADAMTS5
SCHEMBL8240781 0.73 SMN1; SMN2 (0.55) SMN1; SMN2NPSR1ALDH1A1MMP2FPR2
SCHEMBL13792422 0.73 SMN1; SMN2 (0.84) SMN1; SMN2NPSR1ALDH1A1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3103797-B1 2,5-DIOXOIMIDAZOLIDIN-1-YL-3-PHENYLUREA DERIVATIVES AS FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS ALLERGAN INC (US) 2019-04-10 EP disclosed
EP-3103797-A1 2,5-DIOXOIMIDAZOLIDIN-1-YL-3-PHENYLUREA DERIVATIVES AS FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2016-12-14 EP disclosed
EP-2776403-B1 2,5-DIOXOIMIDAZOLIDIN-1-YL-3-PHENYLUREA DERIVATIVES AS FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS ALLERGAN INC (US) 2016-09-14 EP disclosed
US-20130123215-A1 2,5-DIOXOIMIDAZOLIDIN-1-YL-3-PHENYLUREA DERIVATIVES AS FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123215-A1 2,5-DIOXOIMIDAZOLIDIN-1-YL-3-PHENYLUREA DERIVATIVES AS FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS FPR1, FPR2, FPR3 SMN1; SMN2 4512/4885NPSR1 63/4885ALDH1A1 3811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.