SCHEMBL1493722

SCHEMBL1493722

O=c1c(NCC23CC4CC(CC(C4)C2)C3)nn(CCCCC(F)(F)F)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 14/20 0.43
CNR1 P21554 4/20 0.43
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1493643 0.86 CNR2 (0.48) CNR2CNR1HDAC1HDAC6
SCHEMBL1493689 0.77 TLR7 (0.38) CNR2CNR1
SCHEMBL1493630 0.75 AURKA (0.40) CNR2CNR1HDAC1HDAC6KDM4E
SCHEMBL1493640 0.75 CNR2 (0.51) CNR2CNR1
SCHEMBL1491875 0.73 CNR2 (0.39) CNR2CNR1HDAC1HDAC6KDM4E
SCHEMBL13690656 0.66 KDM4E (0.39) CNR2CNR1HDAC1HDAC6KDM4E
SCHEMBL1493624 0.66 AURKA (0.42) CNR2CNR1HDAC1HDAC6KDM4E
SCHEMBL4050608 0.65 CNR1 (0.52) CNR2CNR1HDAC1HDAC6KDM4E
SCHEMBL593602 0.65 LMNA (0.46) CNR2KDM4EALDH1A1LMNANPSR1
SCHEMBL4051371 0.64 CNR1 (0.51) CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011033225-A2 SUBSTITUTED 3-AMINO-CINNOLIN-4(1H)-ONE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-03-24 WO claimed
WO-2011033225-A2 SUBSTITUTED 3-AMINO-CINNOLIN-4(1H)-ONE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-03-24 WO disclosed