SCHEMBL14937490

SCHEMBL14937490

Cc1ccc2ccccc2c1NC=O

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.48
CYP2A6 P11509 3/20 0.48
CYP1A2 P05177 3/20 0.48
ALDH1A1 P00352 4/20 0.42
HSD17B10 Q99714 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
G6PD P11413 1/20 0.38
HPGD P15428 1/20 0.38
ERN1 O75460 1/20 0.38
HCRTR1 O43613 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
HTT P42858 1/20 0.37
S1PR4 O95977 1/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
KCNJ11 Q14654 1/20 0.37
HPRT1 P00492 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798650 0.79 PABPC1 (0.47) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
SCHEMBL1705487 0.78 TSHR (0.58) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
SCHEMBL9806709 0.76 TSHR (0.56) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
SCHEMBL23808919 0.76 KCNJ11 (0.46) TSHRCYP2A6CYP1A2ALDH1A1HKDC1
Hydrochloric Acid SCHEMBL28311925 0.75 TSHR (0.54) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
SCHEMBL23863714 0.75 TSHR (0.54) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL5713244 0.75 TSHR (0.54) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
SCHEMBL18415509 0.74 TSHR (0.48) TSHRCYP2A6CYP1A2ALDH1A1HKDC1
SCHEMBL7415855 0.74 CYP1A2 (0.48) TSHRCYP2A6CYP1A2ALDH1A1HSD17B10
SCHEMBL6374171 0.74 TSHR (0.48) TSHRCYP2A6CYP1A2ALDH1A1HKDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3444031-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2019-02-20 EP disclosed
US-8822724-B2 Method for producing carboxylic acid amide SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2014-09-02 US disclosed
EP-2599769-A1 METHOD FOR PRODUCING CARBOXYLIC ACID AMIDE Sumitomo Chemical Company Limited (JP) 2013-06-05 EP disclosed
US-20130123505-A1 METHOD FOR PRODUCING CARBOXYLIC ACID AMIDE SUMITOMO CHEMICAL COMPANY, LIMITED 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123505-A1 METHOD FOR PRODUCING CARBOXYLIC ACID AMIDE HCAR2, NAAA, FAAH2 TSHR 667/4885CYP2A6 72/4885CYP1A2 25/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.