SCHEMBL14939115

SCHEMBL14939115

Cc1cccc2c1C(=O)C(c1ccccc1)(N1CCN(Cc3cccnc3)CC1)C2=O

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.60
LMNA P02545 1/20 0.47
TRPV6 Q9H1D0 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM3 P20309 1/20 0.44
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 3/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
OPRL1 P41146 1/20 0.42
MAPT P10636 1/20 0.41
P2RX7 Q99572 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939097 0.89 NPSR1 (0.64) NPSR1LMNAKDM4EALDH1A1OPRL1
SCHEMBL14938982 0.88 NPSR1 (0.64) NPSR1LMNATRPV6CHRM2CHRM3
SCHEMBL14939433 0.82 NPSR1 (0.59) NPSR1LMNAKDM4EALDH1A1MAPT
SCHEMBL14939690 0.82 NPSR1 (0.77) NPSR1LMNATRPV6CHRM2CHRM3
SCHEMBL14939022 0.82 NPSR1 (0.59) NPSR1LMNACHRM2CHRM3KDM4E
SCHEMBL14939318 0.80 NPSR1 (0.60) NPSR1TRPV6CHRM2CHRM3KDM4E
SCHEMBL14939850 0.80 NPSR1 (0.60) NPSR1LMNATRPV6CHRM2CHRM3
SCHEMBL14939951 0.79 NPSR1 (0.54) NPSR1LMNAKDM4EALDH1A1MAPT
SCHEMBL14938946 0.78 NPSR1 (0.54) NPSR1LMNAALDH1A1
SCHEMBL14938941 0.78 NPSR1 (0.54) NPSR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed