SCHEMBL14939145

SCHEMBL14939145

COc1ccccc1CN1CCN(C2(c3cc(C)nc(Cl)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.47
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
PHGDH O43175 1/20 0.44
HTT P42858 1/20 0.43
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2B P41595 1/20 0.41
HTR7 P34969 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
TACR2 P21452 1/20 0.40
TACR1 P25103 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939760 0.93 NPSR1 (0.49) NPSR1KDM4EALDH1A1PHGDHHTT
SCHEMBL14940282 0.88 NPSR1 (0.51) NPSR1ALDH1A1PHGDHHTTKMT2A
SCHEMBL14939747 0.88 NPSR1 (0.51) NPSR1KDM4EALDH1A1PHGDHMEN1
SCHEMBL14939586 0.88 NPSR1 (0.51) NPSR1KDM4EALDH1A1PHGDHHTT
SCHEMBL14939314 0.86 NPSR1 (0.47) NPSR1KDM4EALDH1A1MEN1KMT2A
SCHEMBL14940278 0.85 NPSR1 (0.67) NPSR1KDM4EALDH1A1PHGDHHTT
SCHEMBL14939733 0.85 NPSR1 (0.47) NPSR1KDM4EALDH1A1PHGDHHTT
SCHEMBL14938717 0.83 PHGDH (0.52) NPSR1KDM4EALDH1A1PHGDHHTT
SCHEMBL14938994 0.83 NPSR1 (0.47) NPSR1KDM4EALDH1A1HTTMEN1
SCHEMBL14939174 0.83 NPSR1 (0.65) NPSR1KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed