SCHEMBL14939760

SCHEMBL14939760

COc1ccccc1CN1CCN(C2(c3cc(C)nc(C)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.49
PHGDH O43175 1/20 0.47
MEN1 O00255 5/20 0.45
KMT2A Q03164 5/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
HTR2B P41595 1/20 0.45
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
TNKS O95271 1/20 0.43
PARP1 P09874 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
CYP2D6 P10635 2/20 0.43
TSHR P16473 2/20 0.43
HTR7 P34969 1/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939145 0.93 NPSR1 (0.47) NPSR1PHGDHMEN1KMT2AHTR1A
SCHEMBL14939733 0.89 NPSR1 (0.47) NPSR1PHGDHMEN1KMT2AHTR1A
SCHEMBL14938717 0.88 PHGDH (0.52) NPSR1PHGDHMEN1KMT2AHTR1A
SCHEMBL14938994 0.88 NPSR1 (0.47) NPSR1MEN1KMT2AHTR1ADRD2
SCHEMBL14938722 0.87 NPSR1 (0.53) NPSR1PHGDHKMT2AALDH1A1HTT
SCHEMBL14939374 0.87 NPSR1 (0.53) NPSR1PHGDHMEN1KMT2AKDM4E
SCHEMBL14939174 0.87 NPSR1 (0.65) NPSR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL14939609 0.85 NPSR1 (0.52) NPSR1MEN1KMT2AHTR1ADRD2
SCHEMBL14939204 0.85 KDM4E (0.44) NPSR1PHGDHMEN1KMT2AHTR1A
SCHEMBL14939752 0.85 MEN1 (0.55) NPSR1MEN1KMT2AHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed