SCHEMBL14940282

SCHEMBL14940282

CCc1ccccc1CN1CCN(C2(c3cc(C)nc(Cl)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.51
MAPT P10636 4/20 0.42
ADAM17 P78536 2/20 0.39
TP53 P04637 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
ALDH1A1 P00352 2/20 0.35
PHGDH O43175 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
KMT2A Q03164 1/20 0.34
HTR7 P34969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14938722 0.93 NPSR1 (0.53) NPSR1MAPTADAM17TP53LMNA
SCHEMBL14939586 0.92 NPSR1 (0.51) NPSR1MAPTADAM17TP53HTT
SCHEMBL14939747 0.92 NPSR1 (0.51) NPSR1MAPTADAM17TP53LMNA
SCHEMBL14940278 0.89 NPSR1 (0.67) NPSR1MAPTADAM17LMNATSHR
SCHEMBL14939145 0.88 NPSR1 (0.47) NPSR1MAPTHTTALDH1A1PHGDH
SCHEMBL14939726 0.86 NPSR1 (0.47) NPSR1MAPTADAM17TP53LMNA
SCHEMBL14939314 0.85 NPSR1 (0.47) NPSR1MAPTADAM17TP53LMNA
SCHEMBL14939374 0.84 NPSR1 (0.53) NPSR1MAPTADAM17TP53LMNA
SCHEMBL14939879 0.84 NPSR1 (0.53) NPSR1MAPTADAM17TP53LMNA
SCHEMBL14939199 0.84 NPSR1 (0.55) NPSR1MAPTTP53LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed