SCHEMBL14939437

SCHEMBL14939437

COc1ccccc1CN1CCN(C2(c3ccccn3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 4/20 0.48
BCHE P06276 1/20 0.48
HTT P42858 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CCR8 P51685 1/20 0.45
KCNH2 Q12809 1/20 0.45
CYP2D6 P10635 4/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 2/20 0.44
ALOX15 P16050 1/20 0.44
HTR7 P34969 1/20 0.44
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939762 0.88 ALDH1A1 (0.45) ALDH1A1KDM4EBCHEHTTMEN1
SCHEMBL14939260 0.86 NPSR1 (0.49) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL14938959 0.85 NPSR1 (0.48) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL14939204 0.85 KDM4E (0.44) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL14940151 0.84 MEN1 (0.44) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL14939174 0.84 NPSR1 (0.65) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL14939998 0.84 MEN1 (0.45) ALDH1A1KDM4EBCHEHTTMEN1
SCHEMBL14939271 0.83 MEN1 (0.44) ALDH1A1KDM4EBCHEHTTMEN1
SCHEMBL14939213 0.83 MEN1 (0.44) ALDH1A1KDM4EBCHEHTTMEN1
SCHEMBL14939831 0.83 NPSR1 (0.51) ALDH1A1KDM4EHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed