SCHEMBL14939271

SCHEMBL14939271

COc1ccccc1CN1CCN(C2(c3cnc4ccccc4n3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
BCHE P06276 1/20 0.43
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 4/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
CYP2D6 P10635 3/20 0.41
TSHR P16473 2/20 0.41
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2B P41595 1/20 0.41
ALOX15 P16050 1/20 0.41
HTR7 P34969 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939765 0.88 NPSR1 (0.46) ALDH1A1KDM4ENPSR1HTR1A
SCHEMBL14940084 0.87 MEN1 (0.47) MEN1KMT2AL3MBTL1BCHEALDH1A1
SCHEMBL14940355 0.87 HCRTR2 (0.45) MEN1KMT2AKDM4ENPSR1
SCHEMBL14939437 0.83 ALDH1A1 (0.48) MEN1KMT2ABCHEALDH1A1KDM4E
SCHEMBL14939887 0.82 NPSR1 (0.64) ALDH1A1KDM4EHTTNPSR1DRD2
SCHEMBL14939204 0.82 KDM4E (0.44) MEN1KMT2AL3MBTL1ALDH1A1KDM4E
SCHEMBL14940134 0.82 SIGMAR1 (0.51) MEN1KMT2AALDH1A1KDM4ENPSR1
SCHEMBL14940151 0.81 MEN1 (0.44) MEN1KMT2AL3MBTL1ALDH1A1KDM4E
SCHEMBL14939174 0.81 NPSR1 (0.65) MEN1KMT2AALDH1A1KDM4ENPSR1
SCHEMBL14939152 0.80 KDM4E (0.44) MEN1KMT2ABCHEALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed