SCHEMBL14939458

SCHEMBL14939458

COc1cccc(CN2CCN(C3(c4cncc(Br)c4)C(=O)c4ccccc4C3=O)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.52
SIGMAR1 Q99720 1/20 0.50
ALDH1A1 P00352 5/20 0.48
ALDH3A1 P30838 1/20 0.48
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
KDM4E B2RXH2 5/20 0.44
GAA P10253 2/20 0.44
TSHR P16473 2/20 0.44
ALOX15 P16050 1/20 0.44
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
FAAH O00519 1/20 0.43
CHRM2 P08172 1/20 0.42
CHRM3 P20309 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GFER P55789 1/20 0.42
RECQL P46063 1/20 0.42
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939475 0.89 NPSR1 (0.58) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA
SCHEMBL14939432 0.87 NPSR1 (0.68) NPSR1SIGMAR1ALDH1A1LMNAMAPT
SCHEMBL14940026 0.87 NPSR1 (0.56) NPSR1SIGMAR1ALDH1A1ALDH3A1KDM4E
SCHEMBL14939713 0.85 NPSR1 (0.65) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA
SCHEMBL14940106 0.85 NPSR1 (0.72) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA
SCHEMBL14939758 0.84 NPSR1 (0.63) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA
SCHEMBL14939162 0.84 SIGMAR1 (0.51) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA
SCHEMBL14939364 0.83 NPSR1 (0.46) NPSR1ALDH1A1HTTKDM4ETSHR
SCHEMBL14939645 0.82 SIGMAR1 (0.53) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA
SCHEMBL14939975 0.82 NPSR1 (0.60) NPSR1SIGMAR1ALDH1A1ALDH3A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed