SCHEMBL14939432

SCHEMBL14939432

O=C1c2ccccc2C(=O)C1(c1cncc(Br)c1)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.68
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
MAPT P10636 2/20 0.43
TRPC5 Q9UL62 1/20 0.41
SIGMAR1 Q99720 3/20 0.40
DRD2 P14416 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR2B P41595 2/20 0.40
LMNA P02545 1/20 0.39
IGF1R P08069 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939865 0.87 NPSR1 (0.51) NPSR1MAPTSIGMAR1ALDH1A1
SCHEMBL14939458 0.87 NPSR1 (0.52) NPSR1MAPTSIGMAR1DRD2HTR2B
SCHEMBL14939424 0.87 NPSR1 (0.68) NPSR1MMP2MMP9MAPTSIGMAR1
SCHEMBL14940030 0.87 NPSR1 (0.68) NPSR1MMP2MMP9MAPTSIGMAR1
SCHEMBL14939890 0.86 NPSR1 (0.49) NPSR1MAPTTRPC5LMNACYP2D6
SCHEMBL14939297 0.85 NPSR1 (0.48) NPSR1MAPTTRPC5LMNA
SCHEMBL14939840 0.85 NPSR1 (0.77) NPSR1MMP2MMP9MAPTSIGMAR1
SCHEMBL14939690 0.83 NPSR1 (0.77) NPSR1MMP2MMP9MAPTLMNA
SCHEMBL14939364 0.83 NPSR1 (0.46) NPSR1MAPTDRD2HTR2BALDH1A1
SCHEMBL14939617 0.82 NPSR1 (1.00) NPSR1MMP2MMP9MAPTSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed