SCHEMBL14939615

SCHEMBL14939615

Cc1ccc(F)cc1CN1CCN(C2(c3cccc(C(F)(F)F)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
NPSR1 Q6W5P4 1/20 0.47
OPRL1 P41146 3/20 0.42
LMNA P02545 1/20 0.41
HTR7 P34969 1/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
UBE2M P61081 2/20 0.40
DCUN1D1 Q96GG9 2/20 0.40
KDM4E B2RXH2 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TNF P01375 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
SMO Q99835 1/20 0.38
TP53 P04637 1/20 0.38
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939266 0.90 MAPT (0.55) MAPTNPSR1OPRL1HTR7DRD2
SCHEMBL14939190 0.90 MAPT (0.57) MAPTNPSR1OPRL1LMNAHTR7
SCHEMBL14939262 0.90 NPSR1 (0.53) MAPTNPSR1LMNAKDM4ETDP1
SCHEMBL14939138 0.88 NPSR1 (0.51) MAPTNPSR1LMNAHTR7KDM4E
SCHEMBL14939675 0.88 NPSR1 (0.43) MAPTNPSR1LMNAHTR7UBE2M
SCHEMBL14939270 0.88 NPSR1 (0.61) MAPTNPSR1LMNADRD2DRD4
SCHEMBL14939180 0.87 NPSR1 (0.50) MAPTNPSR1LMNAKDM4ETDP1
SCHEMBL14939168 0.87 MAPT (0.53) MAPTNPSR1LMNAHTR7DRD2
SCHEMBL14940182 0.86 NPSR1 (0.45) MAPTNPSR1LMNADRD2KDM4E
SCHEMBL14939636 0.86 MAPT (0.54) MAPTNPSR1LMNAHTR7DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed