SCHEMBL14939712

SCHEMBL14939712

Cc1cccc(C2(N3CCN(Cc4cc(F)ccc4F)CC3)Cc3cc(F)ccc3C2=O)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
MPO P05164 1/20 0.35
HTR6 P50406 2/20 0.35
ALDH1A1 P00352 6/20 0.34
MAPT P10636 1/20 0.34
CHRM4 P08173 1/20 0.33
DPP4 P27487 1/20 0.33
TP53 P04637 1/20 0.33
KDM4E B2RXH2 2/20 0.32
P2RX7 Q99572 1/20 0.32
GAA P10253 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HTT P42858 1/20 0.32
MEN1 O00255 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
DRD2 P14416 2/20 0.32
DRD4 P21917 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939513 0.93 ALDH1A1 (0.36) MPOHTR6ALDH1A1MAPTKDM4E
SCHEMBL14939853 0.92 ALDH1A1 (0.36) BCHEACHEMPOHTR6ALDH1A1
SCHEMBL14939949 0.88 TP53 (0.41) HTR6ALDH1A1MAPTTP53KDM4E
SCHEMBL14939286 0.88 BCHE (0.35) BCHEACHEMPOHTR6ALDH1A1
SCHEMBL14939526 0.88 NPSR1 (0.46) ALDH1A1MAPTKDM4EHTTMEN1
SCHEMBL14940045 0.85 HTR6 (0.38) MPOHTR6ALDH1A1KDM4EGAA
SCHEMBL14939854 0.84 CHRM2 (0.43) ACHEALDH1A1KDM4EHTTDRD2
SCHEMBL14938855 0.83 ALDH1A1 (0.38) MPOHTR6ALDH1A1MAPTTP53
SCHEMBL14940190 0.83 ALDH1A1 (0.37) MPOHTR6ALDH1A1MAPTKDM4E
SCHEMBL14940207 0.82 ALDH1A1 (0.46) ACHEHTR6ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed