SCHEMBL14939853

SCHEMBL14939853

O=C1c2ccc(F)cc2CC1(c1cccc(F)c1)N1CCN(Cc2cc(F)ccc2F)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HTR6 P50406 3/20 0.35
MPO P05164 1/20 0.35
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RIPK1 Q13546 1/20 0.34
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
KDM4E B2RXH2 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CHRM4 P08173 1/20 0.33
SIGMAR1 Q99720 2/20 0.33
SCN9A Q15858 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939712 0.92 BCHE (0.36) ALDH1A1HTR6MPOBCHEACHE
SCHEMBL14940045 0.88 HTR6 (0.38) ALDH1A1HTR6MPONPSR1KDM4E
SCHEMBL14939545 0.87 ALDH1A1 (0.36) ALDH1A1HTR6BCHEACHENPSR1
SCHEMBL14940059 0.87 NPSR1 (0.49) ALDH1A1NPSR1SIGMAR1DRD2HTR2A
SCHEMBL14939513 0.84 ALDH1A1 (0.36) ALDH1A1HTR6MPOKDM4EDRD2
SCHEMBL14939706 0.83 DRD4 (0.44) ALDH1A1KDM4ESMN1; SMN2SIGMAR1DRD2
SCHEMBL14939342 0.82 CYP2D6 (0.48) ALDH1A1HTR6MEN1KMT2ADRD2
SCHEMBL14938855 0.82 ALDH1A1 (0.38) ALDH1A1HTR6MPONPSR1KDM4E
SCHEMBL14940190 0.82 ALDH1A1 (0.37) ALDH1A1HTR6MPONPSR1KDM4E
SCHEMBL14938926 0.82 NPSR1 (0.38) ALDH1A1HTR6MPONPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed