SCHEMBL14940355

SCHEMBL14940355

Cc1ccccc1CN1CCN(C2(c3cnc4ccccc4n3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 3/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KMT2A Q03164 3/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
NPC1 O15118 1/20 0.43
TRPC5 Q9UL62 3/20 0.41
LMNA P02545 4/20 0.40
FABP6 P51161 1/20 0.40
CYP2A13 Q16696 1/20 0.40
HCRTR1 O43613 2/20 0.39
ACHE P22303 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939765 0.90 NPSR1 (0.46) HCRTR2NPSR1RAB9ANPC1HCRTR1
SCHEMBL14939271 0.87 MEN1 (0.44) NPSR1KMT2AMEN1KDM4E
SCHEMBL14940429 0.86 NPSR1 (0.46) NPSR1KMT2ARAB9AMEN1NPC1
SCHEMBL14939887 0.84 NPSR1 (0.64) HCRTR2NPSR1RAB9ANPC1LMNA
SCHEMBL14939324 0.84 NPSR1 (0.48) NPSR1KMT2ARAB9AMEN1NPC1
SCHEMBL14938959 0.82 NPSR1 (0.48) NPSR1KMT2ARAB9AMEN1TRPC5
SCHEMBL14939664 0.82 FABP6 (0.47) NPSR1KMT2ARAB9AMEN1TRPC5
SCHEMBL14939886 0.81 NPSR1 (0.47) NPSR1KMT2ARAB9AMEN1NPC1
SCHEMBL14940304 0.80 NPSR1 (0.46) NPSR1KMT2ARAB9AMEN1NPC1
SCHEMBL14939398 0.80 NPSR1 (0.46) NPSR1KMT2ARAB9AMEN1TRPC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed