SCHEMBL14939765

SCHEMBL14939765

CCc1ccccc1CN1CCN(C2(c3cnc4ccccc4n3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HCRTR2 O43614 12/20 0.38
HCRTR1 O43613 10/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
FAAH O00519 1/20 0.35
ADAM17 P78536 1/20 0.35
HTR1A P08908 1/20 0.35
KCNH2 Q12809 1/20 0.35
LTC4S Q16873 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940355 0.90 HCRTR2 (0.45) NPSR1NPC1RAB9AHCRTR2HCRTR1
SCHEMBL14939271 0.88 MEN1 (0.44) NPSR1KDM4EALDH1A1HTR1A
SCHEMBL14940076 0.86 NPSR1 (0.46) NPSR1NPC1RAB9APOLBFAAH
SCHEMBL14939887 0.85 NPSR1 (0.64) NPSR1NPC1RAB9AHCRTR2HCRTR1
SCHEMBL14939899 0.83 NPSR1 (0.48) NPSR1ADAM17
SCHEMBL14939260 0.82 NPSR1 (0.49) NPSR1KDM4EALDH1A1POLB
SCHEMBL14938910 0.81 NPSR1 (0.46) NPSR1KDM4EALDH1A1
SCHEMBL14939130 0.80 NPSR1 (0.47) NPSR1
SCHEMBL14939940 0.80 NPSR1 (0.47) NPSR1NPC1ADAM17
SCHEMBL14939657 0.79 NPSR1 (0.46) NPSR1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed