SCHEMBL14943015

SCHEMBL14943015

CCCOc1cc(Cl)c2sc(S(=O)(=O)NCP(=O)(O)Oc3ccc(S(=O)(=O)C(F)(F)F)c(F)c3)cc2c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 4/20 0.34
LGALS8 O00214 2/20 0.33
LGALS3 P17931 2/20 0.33
EPAS1 Q99814 1/20 0.31
S1PR4 O95977 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
S1PR5 Q9H228 1/20 0.31
HTT P42858 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13032119 0.94 LGALS8 (0.33) LGALS8LGALS3EPAS1
SCHEMBL14931395 0.90 LGALS8 (0.31) LGALS8LGALS3
SCHEMBL14943011 0.85 TRPV4 (0.38) KAT6A
SCHEMBL14931396 0.84
SCHEMBL14943084 0.81 AR (0.35)
SCHEMBL14943033 0.78
SCHEMBL14943035 0.77 CA2 (0.32)
SCHEMBL3483487 0.76 LGALS8 (0.31) LGALS8LGALS3
SCHEMBL14942993 0.74 EPAS1 (0.31) EPAS1
SCHEMBL3483171 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8440643-B2 Inhibitors of beta-lactamase METHYLGENE INC. (CA) 2013-05-14 US disclosed