SCHEMBL14944647

SCHEMBL14944647

COC(=O)c1cccc(Cn2c3c([nH]c2=O)C(N)N(C)C(n2cccn2)=N3)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.41
OPRD1 P41143 1/20 0.38
ABHD6 Q9BV23 1/20 0.38
IDO1 P14902 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
TPH1 P17752 2/20 0.37
TPH2 Q8IWU9 2/20 0.37
CYP4F2 P78329 2/20 0.37
CYP4A11 Q02928 2/20 0.37
MAPK10 P53779 1/20 0.37
DPP4 P27487 1/20 0.36
P2RX3 P56373 1/20 0.36
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CD74 P04233 1/20 0.35
MIF P14174 1/20 0.35
TRPA1 O75762 1/20 0.35
MAPK8 P45983 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14944673 0.72 TLR7 (0.64) TLR7
SCHEMBL14944713 0.68 ADORA1 (0.35) TLR7HTT
SCHEMBL14987126 0.68 HTT (0.71) ABHD6IDO1LOXL2CYP4F2CYP4A11
SCHEMBL14944715 0.66 TLR7 (0.41) TLR7
SCHEMBL14944714 0.66 TLR7 (0.44) TLR7OPRD1ABHD6IDO1LOXL2
SCHEMBL23997296 0.65 LMNA (0.53) TLR7ABHD6IDO1LOXL2CYP4F2
SCHEMBL30345095 0.65 LMNA (0.53) TLR7ABHD6IDO1LOXL2CYP4F2
SCHEMBL6167291 0.64 TP53 (0.62) MAPTL3MBTL1
SCHEMBL21581161 0.64 TLR7 (0.55) TLR7
SCHEMBL20343835 0.63 TLR7 (0.40) TLR7OPRD1ABHD6IDO1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068438-A1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN R&D IRELAND (IE) 2013-05-16 WO disclosed