SCHEMBL1494522

SCHEMBL1494522

O=C(O)Nc1c(F)ccc(Br)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 4/20 0.36
HTT P42858 2/20 0.36
KIF11 P52732 1/20 0.36
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
IDO1 P14902 3/20 0.33
EGFR P00533 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
HPGD P15428 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
TDO2 P48775 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19331127 0.85 ALDH1A1 (0.38) KMT2AALDH1A1HTTKIF11NPC1
SCHEMBL30262599 0.83 IDO1 (0.43) KMT2AALDH1A1HTTKIF11MEN1
SCHEMBL10129973 0.83 IDO1 (0.43) KMT2AALDH1A1HTTKIF11MEN1
SCHEMBL28439006 0.79 L3MBTL1 (0.44) ALDH1A1HTTRAB9AMAPTSMN1; SMN2
SCHEMBL30387764 0.79 L3MBTL1 (0.44) ALDH1A1HTTRAB9AMAPTSMN1; SMN2
SCHEMBL23043120 0.77 KMT2A (0.49) KMT2AALDH1A1HTTNPC1RAB9A
SCHEMBL3475291 0.77 SLC2A1 (0.42) KMT2AALDH1A1HTTNPC1RAB9A
SCHEMBL20577762 0.77 HDAC1 (0.37) KMT2AALDH1A1NPC1RAB9AMEN1
SCHEMBL20721915 0.76 HDAC1 (0.40) KMT2AALDH1A1NPC1RAB9AMEN1
SCHEMBL6523050 0.75 ATR (0.40) KMT2AHTTNPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470528-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS Novartis AG (CH) 2012-07-04 EP disclosed
WO-2011023773-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS NOVARTIS AG (CH) 2011-03-03 WO disclosed