SCHEMBL14949202

SCHEMBL14949202

COc1ccc2c(Oc3ccc(-c4nnc(Nc5cccc(C)c5)[nH]4)cc3)ncnc2c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 7/20 0.50
EGFR P00533 3/20 0.44
KDR P35968 7/20 0.43
TRPA1 O75762 1/20 0.41
PDGFRB P09619 3/20 0.40
FLT4 P35916 3/20 0.40
FLT3 P36888 3/20 0.40
RAF1 P04049 1/20 0.40
BRAF P15056 1/20 0.40
AURKB Q96GD4 1/20 0.40
RET P07949 1/20 0.39
SRC P12931 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14949334 0.93 CSF1R (0.46) CSF1REGFRKDRTRPA1PDGFRB
SCHEMBL14949213 0.90 EGFR (0.54) CSF1REGFRKDRPDGFRBFLT4
SCHEMBL12336401 0.88 BRAF (0.53) CSF1REGFRKDRFLT3RAF1
SCHEMBL14949214 0.85 KDR (0.49) CSF1RKDRPDGFRBFLT3AURKB
SCHEMBL14949342 0.82 EGFR (0.53) EGFRKDRPDGFRBFLT4RAF1
SCHEMBL14949220 0.82 HTT (0.39) EGFRKDRBRAF
SCHEMBL14949277 0.82 KDR (0.43) EGFRKDR
SCHEMBL12336530 0.81 BRAF (0.50) CSF1REGFRKDRFLT4RAF1
SCHEMBL14949223 0.80 KDR (0.49) KDR
SCHEMBL14949374 0.79 KDR (0.42) EGFRKDRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160096824-A1 Heterocyclic Compounds Useful for Kinase Inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. 2016-04-07 US disclosed
US-9212151-B2 Heterocyclic compounds useful for kinase inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. (US) 2015-12-15 US disclosed
US-20150158828-A1 Heterocyclic Compounds Useful for Kinase Inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. 2015-06-11 US disclosed
US-8957216-B2 Heterocyclic compounds useful for kinase inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. (US) 2015-02-17 US disclosed
US-20130123284-A1 HETEROCYCLIC COMPOUNDS USEFUL FOR KINASE INHIBITION AMITECH THERAPEUTIC SOLUTIONS INC (US) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123284-A1 HETEROCYCLIC COMPOUNDS USEFUL FOR KINASE INHIBITION MAP4K2, MAP3K20, MAP3K19 CSF1R 2451/4885EGFR 499/4885KDR 533/4885
US-20150158828-A1 Heterocyclic Compounds Useful for Kinase Inhibition MAP4K2, MAP3K20, MAP3K19 CSF1R 2451/4885EGFR 499/4885KDR 533/4885
US-20160096824-A1 Heterocyclic Compounds Useful for Kinase Inhibition MAP4K2, MAP3K20, MAP3K19 CSF1R 2451/4885EGFR 499/4885KDR 533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.