SCHEMBL14949680

SCHEMBL14949680

Nc1nc2ccc(Oc3ccc(NC(=O)O)cc3F)nc2s1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MET P08581 12/20 0.44
RAF1 P04049 3/20 0.39
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
KDR P35968 2/20 0.38
EPHX2 P34913 1/20 0.38
MAP4K4 O95819 1/20 0.38
MAPK3 P27361 1/20 0.37
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853481 0.91 EPHX2 (0.41) METABL1BCREPHX2NPC1
SCHEMBL12892609 0.86 BRAF (0.49) METRAF1ABL1BCRMAP4K4
SCHEMBL2855433 0.86 ALDH1A1 (0.40) KDREPHX2NPC1ALDH1A1LMNA
SCHEMBL2857507 0.85 BRAF (0.39) METABL1BCRKDREPHX2
SCHEMBL14949669 0.82 BRAF (0.55) METABL1BCRKDR
SCHEMBL2864471 0.80 BRAF (0.37) METABL1BCRKDREPHX2
SCHEMBL2861313 0.80 KDR (0.49) KDREPHX2NPC1ALDH1A1LMNA
SCHEMBL1259624 0.79 BRAF (0.36) METABL1BCRMAP4K4
SCHEMBL2861678 0.78 BRAF (0.53) KDRMAP4K4NPC1RAB9A
SCHEMBL4314966 0.77 MEN1 (0.53) METRAF1MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445509-B2 Fused heterocyclic derivatives and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-21 US disclosed