SCHEMBL14949669

SCHEMBL14949669

O=C(O)Nc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3n2)c(F)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRAF P15056 6/20 0.55
KDR P35968 14/20 0.52
PDGFRB P09619 1/20 0.52
KIT P10721 1/20 0.52
FLT1 P17948 1/20 0.52
ABL1 P00519 4/20 0.45
BCR P11274 1/20 0.45
MET P08581 4/20 0.44
RIPK1 Q13546 1/20 0.44
RIPK3 Q9Y572 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859325 0.88 KDR (0.53) BRAFKDRPDGFRBKITFLT1
SCHEMBL12892687 0.87 BRAF (0.71) BRAFKDRPDGFRBKITFLT1
SCHEMBL2860133 0.87 KDR (0.55) BRAFKDRPDGFRBKITFLT1
SCHEMBL1259251 0.87 MET (0.55) BRAFKDRPDGFRBKITFLT1
SCHEMBL1258338 0.86 BRAF (0.56) BRAFKDRPDGFRBKITFLT1
SCHEMBL2859622 0.82 KDR (0.72) BRAFKDRPDGFRBKITFLT1
SCHEMBL2855459 0.82 BRAF (0.57) BRAFKDRPDGFRBKITFLT1
SCHEMBL1258993 0.82 BRAF (0.57) BRAFKDRPDGFRBKITFLT1
SCHEMBL14949680 0.82 MET (0.44) KDRABL1BCRMET
SCHEMBL1259902 0.81 MET (0.62) KDRPDGFRBKITFLT1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445509-B2 Fused heterocyclic derivatives and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-21 US disclosed