SCHEMBL14958587

SCHEMBL14958587

CC(C)(C)c1nc2c(-c3ccc(F)cc3)cccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.48
MGAM O43451 3/20 0.48
SI P14410 3/20 0.48
MGAM2 Q2M2H8 3/20 0.48
BRAF P15056 1/20 0.45
CLK2 P49760 2/20 0.44
PARP1 P09874 2/20 0.42
ENPP1 P22413 1/20 0.42
DAPK3 O43293 1/20 0.41
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
ABL1 P00519 1/20 0.41
NTRK1 P04629 1/20 0.41
LCK P06239 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
IGF1R P08069 1/20 0.41
MET P08581 1/20 0.41
PDGFRB P09619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14958588 0.86 CNR2 (0.52) GAAPARP1CNR2MEN1POLB
SCHEMBL14958590 0.86 MGAM (0.50) GAAMGAMSIMGAM2CLK2
SCHEMBL14958589 0.81 GAA (0.51) GAAMGAMSIMGAM2CLK2
SCHEMBL712492 0.80 MGAM (0.55) GAAMGAMSIMGAM2CLK2
SCHEMBL17300893 0.78 GAA (0.46) GAAMGAMSIMGAM2PARP1
SCHEMBL10248490 0.73 MEN1 (0.53) GAAPARP1MEN1POLBMAPT
SCHEMBL6759197 0.73 MGAM (0.50) GAAMGAMSIMGAM2PARP1
SCHEMBL19000985 0.73 L3MBTL1 (0.47) GAAPARP1MEN1POLBMAPT
SCHEMBL18672684 0.72 ALDH1A1 (0.51) GAAPARP1MEN1POLBMAPT
SCHEMBL3968507 0.71 PARP1 (0.44) GAAPARP1MEN1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445473-B2 Heteroaryl-substituted bicyclic Smac mimetics and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-05-21 US disclosed