SCHEMBL14965200

SCHEMBL14965200

CC(C)(C)N1CCC(COCCN2CCOCC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 2/20 0.40
SIGMAR1 Q99720 2/20 0.38
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
KCNH2 Q12809 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
HTR2A P28223 1/20 0.36
SCN1A P35498 1/20 0.36
HTR2B P41595 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN3A Q9NY46 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTR4 Q13639 2/20 0.36
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21933632 0.88 HRH3 (0.33) SIGMAR1HTR2AHTR2BHRH3
SCHEMBL17451649 0.81 CYP1A2 (0.42) CYP2D6CYP1A2SIGMAR1CYP3A4ALDH1A1
SCHEMBL21933629 0.79 HRH3 (0.36) SIGMAR1ALDH1A1MAPK1HTR2AHTR2B
SCHEMBL13741087 0.79 HRH3 (0.43) CYP1A2SIGMAR1TSHRKCNH2ALDH1A1
SCHEMBL21933934 0.78 SIGMAR1 (0.33) SIGMAR1HTR2AHTR2BHRH3
SCHEMBL16293179 0.78 RECQL (0.54) SMN1; SMN2USP2
SCHEMBL24856304 0.77 HRH3 (0.32) HRH3
SCHEMBL13741195 0.77 HRH3 (0.40) CYP1A2SIGMAR1TSHRKCNH2ALDH1A1
SCHEMBL19370316 0.77 TDP1 (0.40) CYP2D6CYP1A2SIGMAR1TSHRKCNH2
SCHEMBL21025893 0.76 DRD2 (0.33) SIGMAR1ALDH1A1HTR2AHTR2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780343-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS Xention Limited (GB) 2014-09-24 EP disclosed
WO-2013072694-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS XENTION LIMITED (GB) 2013-05-23 WO disclosed