SCHEMBL14965730

SCHEMBL14965730

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1cccc(-c3cccc(F)c3)n1)CC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.37
HTR1A P08908 1/20 0.37
CXCR4 P61073 1/20 0.35
PIK3R1 P27986 4/20 0.35
PIK3CA P42336 4/20 0.35
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
SLC2A1 P11166 1/20 0.34
KCNH2 Q12809 4/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
CACNA1C Q13936 1/20 0.32
SCN5A Q14524 1/20 0.32
ALDH1A1 P00352 2/20 0.32
SCN9A Q15858 1/20 0.32
CHRM1 P11229 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965410 0.87 DRD2 (0.38) DRD2DRD4DRD3SLC2A1KCNH2
SCHEMBL14966131 0.86 DRD2 (0.49) DRD2HTR1ADRD4DRD3SLC2A1
SCHEMBL14965746 0.85 DRD2 (0.41) DRD2DRD4DRD3SLC2A1KCNH2
SCHEMBL14965683 0.85 DRD2 (0.43) DRD2HTR1ADRD4DRD3KCNH2
SCHEMBL14965749 0.85 CYP11B1 (0.43) DRD2DRD4DRD3ALDH1A1CHRM1
SCHEMBL14966129 0.85 SCN9A (0.37) DRD2HTR1ACXCR4SLC2A1KCNH2
SCHEMBL14965655 0.84 PDE4B (0.36) DRD2DRD4DRD3SLC2A1ADORA2A
SCHEMBL14966064 0.83 JAK2 (0.34) DRD2HTR1APIK3R1PIK3CAALDH1A1
SCHEMBL14966011 0.83 MTOR (0.37) DRD2HTR1APIK3R1PIK3CAKCNH2
SCHEMBL14966353 0.83 JAK2 (0.37) DRD2HTR1AKCNH2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed