SCHEMBL14966129

SCHEMBL14966129

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1cccc(-c3ccc(C(F)(F)F)cc3)n1)CC2

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.37
KCNH2 Q12809 3/20 0.36
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
TRPV3 Q8NET8 8/20 0.36
MCHR1 Q99705 1/20 0.36
CHRM1 P11229 1/20 0.35
SLC2A1 P11166 1/20 0.35
CXCR4 P61073 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965897 0.86 HTR1A (0.35) KCNH2HTR1ADRD2SLC2A1CXCR4
SCHEMBL14965895 0.86 HTR1A (0.35) KCNH2HTR1ADRD2SLC2A1CXCR4
SCHEMBL14965893 0.86 SCN9A (0.37) SCN9AKCNH2HTR1ADRD2MCHR1
SCHEMBL14965750 0.85 CHKA (0.43) KCNH2CHRM1SLC2A1
SCHEMBL14965894 0.85 HIF1A (0.41) KCNH2MCHR1CHRM1SLC2A1
SCHEMBL14965730 0.85 DRD2 (0.37) SCN9AKCNH2HTR1ADRD2CHRM1
SCHEMBL14965837 0.84 HIF1A (0.44) KCNH2CHRM1
SCHEMBL14965932 0.83 HIF1A (0.41) CHRM1
SCHEMBL14966162 0.83 CHRM1 (0.36) KCNH2HTR1ADRD2CHRM1
SCHEMBL14971086 0.82 ALDH1A1 (0.41) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed