SCHEMBL14966211

SCHEMBL14966211

CCNC(=O)c1ccc(-c2cc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)ccn2)cc1F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.38
PARP1 P09874 1/20 0.36
TNK1 Q13470 1/20 0.36
MCHR1 Q99705 1/20 0.34
MET P08581 3/20 0.34
CHRM4 P08173 2/20 0.34
HSP90AA1 P07900 2/20 0.33
HSP90AB1 P08238 2/20 0.33
KCNH2 Q12809 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
HDAC1 Q13547 1/20 0.33
MLLT1 Q03111 2/20 0.32
PIK3CA P42336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965574 0.91 HDAC4 (0.36) MCHR1METTBK1HDAC1MLLT1
SCHEMBL14965597 0.90 MTOR (0.39) MTORPARP1TNK1MCHR1MET
SCHEMBL14965517 0.89 FGFR1 (0.40) PARP1TNK1MET
SCHEMBL14965666 0.88 LRRK2 (0.36) METTBK1
SCHEMBL14965835 0.87 MTOR (0.37) MTORPIK3CA
SCHEMBL14965806 0.86 MET (0.39) MTORMETPIK3CA
SCHEMBL14965762 0.86 MTOR (0.39) MTORMETCHRM4HSP90AA1HSP90AB1
SCHEMBL14965970 0.84 MTOR (0.39) MTORMCHR1HSP90AA1HSP90AB1KCNH2
SCHEMBL14966019 0.84 MCHR1 (0.39) MTORMCHR1CHRM4HSP90AA1HSP90AB1
SCHEMBL14966035 0.82 MCHR1 (0.42) PARP1TNK1MCHR1METCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed