SCHEMBL14965776

SCHEMBL14965776

CC(C)(C)OC(=O)CN1CCOc2nc([N+](=O)[O-])cn2CC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.42
PTGS1 P23219 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
CHRM1 P11229 1/20 0.34
CACNA1C Q13936 1/20 0.34
SCN5A Q14524 1/20 0.34
MITF O75030 1/20 0.33
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965833 0.86 KCNH2 (0.41) KCNH2PTGS1SLC6A2SLC6A4CHRM1
SCHEMBL14965729 0.83 KCNH2 (0.42) KCNH2PTGS1SLC6A2SLC6A4CHRM1
SCHEMBL14965944 0.82 KCNH2 (0.37) KCNH2CHRM1MITFALDH1A1LMNA
SCHEMBL14966362 0.76 KCNH2 (0.39) KCNH2PTGS1SLC6A2SLC6A4CHRM1
SCHEMBL5539141 0.76 KCNH2 (0.53) KCNH2PTGS1SLC6A2SLC6A4CHRM1
SCHEMBL14965638 0.76 KCNH2 (0.40) KCNH2PTGS1SLC6A2SLC6A4CHRM1
SCHEMBL5543048 0.72 KCNH2 (0.53) KCNH2PTGS1SLC6A2SLC6A4CACNA1C
SCHEMBL5543143 0.71 KCNH2 (0.55) KCNH2PTGS1SLC6A2SLC6A4CACNA1C
SCHEMBL5543139 0.71 KCNH2 (0.55) KCNH2PTGS1SLC6A2SLC6A4CACNA1C
SCHEMBL3466176 0.70 KCNH2 (0.52) KCNH2PTGS1SLC6A2SLC6A4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed