SCHEMBL14965833

SCHEMBL14965833

CC1(C)Cn2cc([N+](=O)[O-])nc2OCCN1CC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.41
CACNA1C Q13936 1/20 0.36
SCN5A Q14524 1/20 0.36
PTGS1 P23219 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
CHRM1 P11229 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LMNA P02545 1/20 0.32
KMT2A Q03164 3/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
MITF O75030 1/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
SLC6A9 P48067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965776 0.86 KCNH2 (0.42) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL14966362 0.83 KCNH2 (0.39) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL14965638 0.79 KCNH2 (0.40) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL14965582 0.78 HSD17B10 (0.38) KCNH2CHRM1L3MBTL1LMNAKMT2A
SCHEMBL14965729 0.77 KCNH2 (0.42) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL1046316 0.74 CHRM1 (0.40) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL5536536 0.73 KCNH2 (0.53) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL14965864 0.72 ITGB3 (0.39) KCNH2CHRM1LMNAKMT2AALDH1A1
SCHEMBL5543648 0.71 KCNH2 (0.40) KCNH2CACNA1CSCN5APTGS1SLC6A2
SCHEMBL14965869 0.70 ALDH1A1 (0.41) KCNH2CHRM1LMNAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed