SCHEMBL14965879

SCHEMBL14965879

Nc1ccc2cnn(CC(F)(F)F)c(=O)c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
CNR1 P21554 1/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
MITF O75030 1/20 0.35
PKM P14618 1/20 0.35
SRC P12931 1/20 0.35
AURKA O14965 3/20 0.34
SYK P43405 1/20 0.34
AURKB Q96GD4 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
CHEK1 O14757 2/20 0.33
AR P10275 1/20 0.33
KMT2A Q03164 1/20 0.33
DAPK3 O43293 1/20 0.33
CSNK1A1 P48729 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30896807 0.80 HTR2A (0.42) SRCAURKAKDM4ECHEK1DAPK3
SCHEMBL14966684 0.80 GLS (0.45) PTGS2ALDH1A1KMT2APOLB
SCHEMBL22101196 0.75 PTGS2 (0.39) PTGS2TDP1CNR1NPC1RAB9A
SCHEMBL22101239 0.75 NPC1 (0.43) PTGS2TDP1CNR1NPC1RAB9A
SCHEMBL5863967 0.75 TDP1 (0.56) TDP1CNR1PKMAURKAALDH1A1
SCHEMBL14965798 0.75 BRD4 (0.43) PTGS2TDP1NPC1RAB9AMITF
SCHEMBL22393580 0.73 BTK (0.39) PTGS2TDP1CNR1AURKASYK
SCHEMBL22101777 0.73 TDP1 (0.40) PTGS2TDP1CNR1NPC1RAB9A
SCHEMBL14966308 0.73 MAPT (0.44) PKMKMT2APOLB
SCHEMBL14966121 0.72 BRD4 (0.46) PTGS2RAB9APKMALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072825-A1 PHTALAZINONE DERIVATIVES AS MPEGS -1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-05-23 WO disclosed