SCHEMBL14965798

SCHEMBL14965798

Nc1ccc2cnn(CC3CC3)c(=O)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.43
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
NPBWR1 P48145 1/20 0.38
ADORA2A P29274 3/20 0.38
PTGS2 P35354 2/20 0.38
PKM P14618 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A2 O94788 1/20 0.36
ALDH1A3 P47895 1/20 0.36
KAT2B Q92831 1/20 0.36
MERTK Q12866 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
MET P08581 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966121 0.93 BRD4 (0.46) BRD4NPBWR1ADORA2APTGS2PKM
SCHEMBL3387257 0.81 BRD4 (0.48) BRD4HDAC1HDAC2PKM
SCHEMBL14966246 0.80 GLS (0.44) BRD4PTGS2PDE4A
SCHEMBL5863449 0.80 ALDH1A1 (0.48) ALDH1A1KDM4EHSD17B10NPC1RAB9A
SCHEMBL27083872 0.78 HDAC1 (0.51) BRD4HDAC1HDAC2ADORA2APKM
SCHEMBL14965879 0.75 PTGS2 (0.37) PTGS2PKMALDH1A1TDP1KDM4E
SCHEMBL14965797 0.75 CNR2 (0.42) BRD4NPBWR1PTGS2PDE1APDE1B
SCHEMBL5863967 0.74 TDP1 (0.56) BRD4PKMALDH1A1TDP1KDM4E
SCHEMBL20325546 0.72 HDAC1 (0.47) BRD4HDAC1HDAC2NPBWR1ADORA2A
SCHEMBL14965757 0.72 KDM4E (0.40) ALDH1A1TDP1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072825-A1 PHTALAZINONE DERIVATIVES AS MPEGS -1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-05-23 WO disclosed
WO-2013072825-A1 PHTALAZINONE DERIVATIVES AS MPEGS -1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-05-23 WO disclosed