SCHEMBL14966248

SCHEMBL14966248

O=C(Nc1ccc(OC(F)(F)F)cc1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.51
EPAS1 Q99814 1/20 0.51
CHRM1 P11229 1/20 0.49
KCNH2 Q12809 5/20 0.47
ABL1 P00519 1/20 0.47
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MITF O75030 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP2C9 P11712 1/20 0.41
TNF P01375 1/20 0.41
NOD2 Q9HC29 1/20 0.41
NOD1 Q9Y239 1/20 0.41
PRKAA2 P54646 2/20 0.40
CSF1R P07333 1/20 0.40
FLT3 P36888 1/20 0.40
EPHX2 P34913 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
SAE1 Q9UBE0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965959 0.92 KCNH2 (0.53) HIF1AEPAS1CHRM1KCNH2ABL1
SCHEMBL14966147 0.92 KCNH2 (0.53) HIF1AEPAS1CHRM1KCNH2ABL1
SCHEMBL14965787 0.91 HIF1A (0.44) HIF1AEPAS1CHRM1KCNH2ABL1
SCHEMBL14965842 0.87 CHRM1 (0.59) CHRM1KCNH2ABL1SMN1; SMN2
SCHEMBL14965916 0.86 ABL1 (0.56) HIF1AEPAS1CHRM1KCNH2ABL1
SCHEMBL14966083 0.85 CHRM1 (0.52) HIF1AEPAS1CHRM1KCNH2ABL1
SCHEMBL14965624 0.85 CHRM1 (0.57) CHRM1KCNH2
SCHEMBL14965964 0.84 HIF1A (0.52) HIF1AEPAS1MEN1KMT2ASMN1; SMN2
SCHEMBL14966124 0.84 CHRM1 (0.54) CHRM1KCNH2ABL1RAB9A
SCHEMBL14965737 0.84 CHRM1 (0.49) CHRM1KCNH2ABL1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed