SCHEMBL14967451

SCHEMBL14967451

CC(=O)CC1CCC(Oc2ncc(-c3ccc(C=O)c(F)c3)cn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.41
DGAT1 O75907 6/20 0.41
KCNH2 Q12809 6/20 0.41
ADORA2A P29274 2/20 0.41
SOAT1 P35610 3/20 0.38
FFAR4 Q5NUL3 5/20 0.37
ACACB O00763 6/20 0.37
MELK Q14680 1/20 0.37
ERN1 O75460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14968064 0.90 ALDH1A1 (0.40) GRIN2BDGAT1KCNH2ADORA2ASOAT1
SCHEMBL14971854 0.85 ERN1 (0.38) GRIN2BDGAT1KCNH2ADORA2AACACB
SCHEMBL14967450 0.82 ERN1 (0.35) GRIN2BFFAR4ACACBMELKERN1
SCHEMBL14969248 0.81 CYP11B1 (0.38) GRIN2BDGAT1KCNH2ADORA2AFFAR4
SCHEMBL14969247 0.81 CYP11B1 (0.38) GRIN2BDGAT1KCNH2ADORA2AFFAR4
SCHEMBL14969513 0.80 ALDH1A1 (0.40) GRIN2BDGAT1FFAR4MELKERN1
SCHEMBL14969514 0.80 ALDH1A1 (0.40) GRIN2BDGAT1FFAR4MELKERN1
SCHEMBL14968128 0.80 MAPT (0.36) GRIN2BFFAR4ERN1
SCHEMBL14971569 0.79 DGAT1 (0.51) GRIN2BDGAT1KCNH2ADORA2ASOAT1
SCHEMBL15055224 0.79 DGAT1 (0.51) GRIN2BDGAT1KCNH2ADORA2ASOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed