SCHEMBL14969048

SCHEMBL14969048

CC(NS(=O)(=O)c1cccs1)c1nc2nc(N)c(C(N)=O)cc2cc1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
MAPT P10636 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 4/20 0.35
GAA P10253 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCR4 P51679 1/20 0.34
MMP1 P03956 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969189 0.82 IKBKB (0.35) ALDH1A1GAAKDM4EHPGD
SCHEMBL14969297 0.79 ACLY (0.36) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL14969324 0.77 CHRM2 (0.30)
SCHEMBL14969233 0.73 IKBKB (0.40) ALDH1A1GAAKDM4EHPGD
SCHEMBL14969015 0.69 KDM4E (0.39) ALDH1A1GAAKDM4EHPGD
SCHEMBL3140166 0.66 SLC1A3 (0.57) SLC1A3SLC1A2SLC1A1MAPTCYP1A2
SCHEMBL14968966 0.63 IKBKB (0.41) ALDH1A1GAAKDM4EHPGDL3MBTL1
SCHEMBL7915450 0.62 CYP2D6 (0.56) SLC1A3SLC1A2SLC1A1MAPTCYP2C9
SCHEMBL30856551 0.62 SLC1A3 (0.62) SLC1A3SLC1A2SLC1A1CYP2C9CYP2C19
SCHEMBL14969065 0.60 IKBKB (0.41) ALDH1A1GAAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed