SCHEMBL14969189

SCHEMBL14969189

CC(NS(C)(=O)=O)c1nc2nc(N)c(C(N)=O)cc2cc1Br

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969048 0.82 SLC1A3 (0.38) KDM4EALDH1A1GAAHPGD
SCHEMBL14969297 0.81 ACLY (0.36) IKBKBALDH1A1HPGD
SCHEMBL14969324 0.81 CHRM2 (0.30)
SCHEMBL14969233 0.81 IKBKB (0.40) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969015 0.77 KDM4E (0.39) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14968966 0.70 IKBKB (0.41) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969065 0.67 IKBKB (0.41) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969098 0.64 RCE1 (0.36) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL14969185 0.64 RCE1 (0.38) IKBKBKDM4EALDH1A1GLAGAA
SCHEMBL31692851 0.62 IKBKB (0.46) IKBKBKDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed