SCHEMBL14969203

SCHEMBL14969203

CCOC(=O)C1CC(Oc2ncc(-c3ccc(-c4nc5ccccc5[nH]4)c(F)c3)cn2)C1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
FASN P49327 3/20 0.42
DGAT1 O75907 3/20 0.41
DHODH Q02127 5/20 0.40
KCNH2 Q12809 2/20 0.40
ADORA2A P29274 1/20 0.40
NPC1 O15118 3/20 0.38
PKM P14618 3/20 0.38
RAB9A P51151 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HSP90AA1 P07900 1/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969335 0.88 DGAT1 (0.40) ALDH1A1KDM4EDGAT1KCNH2ADORA2A
SCHEMBL14972249 0.88 DGAT1 (0.49) ALDH1A1FASNDGAT1DHODHKCNH2
SCHEMBL14969110 0.88 DGAT1 (0.49) ALDH1A1FASNDGAT1DHODHKCNH2
SCHEMBL14971564 0.84 DGAT1 (0.51) ALDH1A1FASNDGAT1DHODHKCNH2
SCHEMBL14971856 0.81 DGAT1 (0.61) FASNDGAT1KCNH2ADORA2A
SCHEMBL14971761 0.81 DGAT1 (0.61) FASNDGAT1KCNH2ADORA2A
SCHEMBL14968362 0.79 DGAT1 (0.44) DGAT1DHODHKCNH2ADORA2A
SCHEMBL14972233 0.79 DGAT1 (0.45) DGAT1DHODHKCNH2ADORA2A
SCHEMBL14968128 0.79 MAPT (0.36) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL14972187 0.78 DGAT1 (0.59) DGAT1DHODHKCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed