SCHEMBL14969335

SCHEMBL14969335

CCOC(=O)C1CC(Oc2ncc(-c3ccc(-c4nc5cc(C(F)(F)F)ccc5[nH]4)c(F)c3)cn2)C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 14/20 0.40
KCNH2 Q12809 4/20 0.39
SOAT1 P35610 2/20 0.39
ADORA2A P29274 2/20 0.38
SYK P43405 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
AGPAT2 O15120 1/20 0.36
NPBWR1 P48145 1/20 0.35
SSTR2 P30874 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14971563 0.89 DGAT1 (0.47) DGAT1KCNH2SOAT1ADORA2ANPBWR1
SCHEMBL14971609 0.89 DGAT1 (0.47) DGAT1KCNH2SOAT1ADORA2ANPBWR1
SCHEMBL14969219 0.89 DGAT1 (0.47) DGAT1KCNH2SOAT1ADORA2ANPBWR1
SCHEMBL14969203 0.88 ALDH1A1 (0.45) DGAT1KCNH2ADORA2AKDM4ENPC1
SCHEMBL14969256 0.87 DGAT1 (0.45) DGAT1KCNH2SOAT1ADORA2A
SCHEMBL14971708 0.86 DHODH (0.39) DGAT1KCNH2SOAT1ADORA2ANPBWR1
SCHEMBL14971669 0.85 DGAT1 (0.49) DGAT1KCNH2SOAT1ADORA2A
SCHEMBL14971556 0.85 DGAT1 (0.56) DGAT1KCNH2SOAT1ADORA2A
SCHEMBL14970260 0.83 DGAT1 (0.41) DGAT1KCNH2SOAT1ADORA2A
SCHEMBL14971831 0.83 DGAT1 (0.37) DGAT1KCNH2SOAT1ADORA2AAGPAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed